期刊: TETRAHEDRON LETTERS, 2021; 69 ()
Six 6-chlorine-containing briarane analogues, including two new compounds, briarenols U (1) and V (2), as well as four known metabolites, solenolides ......
期刊: TETRAHEDRON LETTERS, 2021; 72 ()
A Rh(III)-catalyzed regioselective C-H nitrosation/annulation reaction of unsymmetrical azobenzenes with [NO][BF4] has been developed to achieve high-......
期刊: TETRAHEDRON LETTERS, 2021; 73 ()
Scopariusicide C (1), a novel ent-clerodane-based meroditerpenoid was isolated from artificially cultivated Isodon scoparius. An oxygen insertion reac......
期刊: TETRAHEDRON LETTERS, 2021; 77 ()
An atom-economical and efficient method for synthesizing 4-organylselanyl-1H-pyrazoles through electrochemical cross-dehydrogenation coupling of N-uns......
期刊: TETRAHEDRON LETTERS, 2021; 78 ()
A practical 1,3-dipolar [3 + 2] cycloaddition of N-2,2,2-trifluoroethylisatin ketimines and (Z)-4-((chro-mone-3-yl)methylene)oxazolones under phase-tr......
期刊: TETRAHEDRON LETTERS, 2021; 79 ()
Antimicrobial peptides are an important part of the natural immune system. According to reports, the antimicrobial peptide piscidins have a very signi......
期刊: TETRAHEDRON LETTERS, 2021; 71 ()
To improve drug efficiency and reduce side effects in cancer therapy, precision therapy with small molecular prodrugs is urgently needed. Podophylloto......
期刊: TETRAHEDRON LETTERS, 2021; 70 ()
A solvent-dependent I-2-catalyzed chemoselective reaction was developed for the synthesis of benzimidazoles and 1,3,5-triarylbenzenes via the annulati......
期刊: TETRAHEDRON LETTERS, 2021; 72 ()
The asymmetric version of Pd(II)/bipyridine-catalyzed nucleophilic addition of arylboronic acids to N-sulfonyl arylaldimines was developed, and excell......
期刊: TETRAHEDRON LETTERS, 2021; 76 ()
An efficient catalytic asymmetric [3 + 2] cyclization of 3-substituted indoles with p-benzoquinones has been realized using a binol-chiral phosphoric ......
期刊: TETRAHEDRON LETTERS, 2021; 78 ()
A copper catalyzed aerobic sp(3) C-H amination of 3,4-dihydroquinoxalin-2(1H)-ones is developed. This protocol provides a concise method to access 3-a......
期刊: TETRAHEDRON LETTERS, 2021; 70 ()
A cobalt-catalyzed C-H activation/cyclization of N-carbamoyl indole/benzamides with maleimides assisted by pyridinylmethylamine under mild reaction co......
期刊: TETRAHEDRON LETTERS, 2021; 72 ()
A copper-catalyzed intramolecular radical cascade acyl-cyanation to synthesize cyano-containing chroman-4-ones has been developed. A series of CN-subs......
期刊: TETRAHEDRON LETTERS, 2021; 72 ()
We described herein a Rh(III)-catalyzed C7-selective C-H activation/annulation of indolines with 1,3-enynes to efficiently access various privileged 1......
期刊: TETRAHEDRON LETTERS, 2021; 73 ()
A catalyst- and additive-free ring-opening polymerization of tetrahydrofuran initiated by phenyl(trifluoroethyl)iodonium triflate ([PhICH2CF3][OTf]) w......